Signal transduction via Ras.

A Wittinghofer
Author Information
  1. A Wittinghofer: Max-Planck-Institut für molekulare Physiologie, Dortmund, Germany.

Abstract

Ras is a major regulator of cell growth. It is a GTP-binding protein that functions as a molecular switch, cycling between the GDP-bound OFF and GTP-bound ON states. In the GTP-bound state it interacts with effector proteins that mediate the biological function. It is found as an oncogene in about 30% of human tumors. Structural and mechanistic studies on Ras and its interaction with effectors and GAP will be discussed in the context of the biology and pathophysiology of this protein.

MeSH Term

Arginine
Catalytic Domain
Enzyme Activation
GTP Phosphohydrolases
GTPase-Activating Proteins
Humans
Hydrolysis
Protein Binding
Proteins
Signal Transduction
ras GTPase-Activating Proteins
ras Proteins

Chemicals

GTPase-Activating Proteins
Proteins
ras GTPase-Activating Proteins
Arginine
GTP Phosphohydrolases
ras Proteins

Word Cloud

Created with Highcharts 10.0.0RasproteinGTP-boundmajorregulatorcellgrowthGTP-bindingfunctionsmolecularswitchcyclingGDP-boundOFFONstatesstateinteractseffectorproteinsmediatebiologicalfunctionfoundoncogene30%humantumorsStructuralmechanisticstudiesinteractioneffectorsGAPwilldiscussedcontextbiologypathophysiologySignaltransductionvia

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