Glaucopines A and B, new cyathane diterpenes from the fruiting bodies of Sarcodon glaucopus.

Massimo Curini, Federica Maltese, Maria Carla Marcotullio, Luigi Menghini, Rita Pagiotti, Ornelio Rosati, Gianmario Altinier, Aurelia Tubaro
Author Information
  1. Massimo Curini: Dipartimento di Chimica e Tecnologia del Farmaco, Sez. Chimica Organica, Università degli Studi, Perugia, Italy.

Abstract

Glaucopine A (1) and B (2), two new cyathane diterpenes, have been isolated from the mushroom Sarcodon glaucopus: their structures have been determined on the basis of spectral data. Their topical anti-inflammatory activity was evaluated using the Croton oil ear test in mice: compounds 1 and 2 (1 micromol/cm2) provoked edema reduction (62 % and 55 %, respectively) similar to that induced by the reference non-steroidal anti-inflammatory drug, indomethacin (0.3 micromol/cm2, 61 % edema reduction).

MeSH Term

Animals
Anti-Inflammatory Agents, Non-Steroidal
Basidiomycota
Croton Oil
Diterpenes
Edema
Fruit
Male
Mice
Mice, Inbred Strains
Phytotherapy
Plant Extracts

Chemicals

Anti-Inflammatory Agents, Non-Steroidal
Diterpenes
Plant Extracts
cyathane
Croton Oil

Word Cloud

Created with Highcharts 10.0.01%B2newcyathanediterpenesSarcodonanti-inflammatorymicromol/cm2edemareductionGlaucopinetwoisolatedmushroomglaucopus:structuresdeterminedbasisspectraldatatopicalactivityevaluatedusingCrotonoileartestmice:compoundsprovoked6255respectivelysimilarinducedreferencenon-steroidaldrugindomethacin0361Glaucopinesfruitingbodiesglaucopus

Similar Articles

Cited By (1)