Quo Vadis after AEGIS: New Opportunities for Therapies Targeted at Reverse Cholesterol Transport?

Nick S R Lan, Gerald F Watts
Author Information
  1. Nick S R Lan: Medical School, The University of Western Australia, Crawley, Perth, Australia.
  2. Gerald F Watts: Medical School, The University of Western Australia, Crawley, Perth, Australia. gerald.watts@uwa.edu.au.

Abstract

PURPOSE OF REVIEW: High-density lipoprotein (HDL) is integral to reverse cholesterol transport (RCT), a process considered to protect against atherosclerotic cardiovascular disease (ASCVD). We summarise findings from the recent AEGIS-II trial and discuss new opportunities for HDL therapeutics targeted at RCT.
RECENT FINDINGS: Mendelian randomisation studies have suggested a causal association between the functional properties of HDL and ASCVD. However, the AEGIS-II trial of CSL112, an apolipoprotein A-I therapy that enhances cholesterol efflux, did not meet its primary endpoint. Exploratory analyses demonstrated that CSL112 significantly reduced ASCVD events among participants with a baseline low-density lipoprotein (LDL)-cholesterol ≥ 100 mg/dL, suggesting that RCT may depend on LDL-cholesterol levels. The role of HDL therapeutics in patients with familial hypercholesterolaemia, inherited low HDL-cholesterol and impaired HDL function, especially with inadequately controlled LDL-cholesterol, merits further investigation. The treatment of patients with monogenic defects in HDL metabolism remains a significant gap in care that needs further research.

Keywords

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MeSH Term

Humans
Atherosclerosis
Biological Transport
Cholesterol
Cholesterol, LDL
Cholesterol, HDL
Apolipoprotein A-I

Chemicals

Cholesterol
Cholesterol, LDL
Cholesterol, HDL
Apolipoprotein A-I

Word Cloud

Created with Highcharts 10.0.0HDLRCTASCVDlipoproteincholesteroldiseaseAEGIS-IItrialtherapeuticsCSL112therapyLDL-cholesterolpatientsCholesterolPURPOSEOFREVIEW:High-densityintegralreversetransportprocessconsideredprotectatheroscleroticcardiovascularsummarisefindingsrecentdiscussnewopportunitiestargetedRECENTFINDINGS:MendelianrandomisationstudiessuggestedcausalassociationfunctionalpropertiesHoweverapolipoproteinA-IenhanceseffluxmeetprimaryendpointExploratoryanalysesdemonstratedsignificantlyreducedeventsamongparticipantsbaselinelow-densityLDL-cholesterol ≥ 100 mg/dLsuggestingmaydependlevelsrolefamilialhypercholesterolaemiainheritedlowHDL-cholesterolimpairedfunctionespeciallyinadequatelycontrolledmeritsinvestigationtreatmentmonogenicdefectsmetabolismremainssignificantgapcareneedsresearchQuoVadisAEGIS:NewOpportunitiesTherapiesTargetedReverseTransport?CardiovasculardiseasesCoronaryarteryDyslipidaemiaLipid-loweringRiskfactors

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