Intestinal absorption and metabolism of a soluble flavonoid, alphaG-rutin, in portal cannulated rats.

Mgumi Matsumoto, Hideyuki Chiji, Hiroshi Hara
Author Information
  1. Mgumi Matsumoto: Fuji Women's University, Faculty of Human Life Science, Department of Food Science and Human Nutrition, Ishikari, Hokkaido, 061-3204, Japan.

Abstract

A highly soluble Quercetin glycoside, alphaG-rutin, is a glucose adduct of insoluble rutin, and intestinal absorption and metabolism of alphaG-rutin has not been known. We investigated the intestinal absorption and metabolism of alphaG-rutin by using portal and duodenal cannulated rats and the isolated rat intestinal mucosa. After a duodenal instillation of alphaG-rutin (150 mumol), intact alphaG-rutin, rutin and Quercetin were appeared in the portal blood and these concentrations were similarly increased at 15 min. Portal Quercetin reached a peak value at 60 min, and the value was higher than those of alphaG-rutin and rutin at that time. Quercetin-conjugates were also increased 30 min after the instillation. The remaining of alphaG-rutin metabolites, mainly rutin, in the intestine were 58% of instilled alphaG-rutin after 150 min. In the experiment by using the isolated mucosa of the jejunum, ileum and cecum, alphaG-rutin and rutin, but not Quercetin, appeared in the serosal sides of all segments, and they were increased linearly from 10 to 100 mmol/l of mucosal alphaG-rutin. We also showed portal injected alphaG-rutin was very rapidly cleared from the blood, and appeared a large amount of conjugates. In conclusion, a soluble flavonoid-glycoside, alphaG-rutin, was absorbed as glycosides into the portal blood. A part of alphaG-rutin was hydrolyzed to rutin, but not to aglycone, through the intestine.

MeSH Term

Animals
Biological Transport
Catheterization
Epithelium
Hydrolysis
Intestinal Absorption
Intestinal Mucosa
Male
Molecular Structure
Portal Vein
Rats
Rats, Wistar
Rutin
Trisaccharides

Chemicals

Trisaccharides
4(G)-alpha-glucopyranosyl-rutin
Rutin

Word Cloud

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