[The current role of isavuconazole in the treatment of invasive fungal infections].

Ondrej Zahornacky, Pavol Jar��u��ka
Author Information
  1. Ondrej Zahornacky: Clinic of Infectology and Travel Medicine, Faculty of Medicine, University of Pavel Jozef ��af��rik and UNLP, Ko��ice, Slovak Republic, e-mail: ondrejzahornacky@gmail.com.

Abstract

Significant medical advances in the treatment and management of immunocompromised patients are currently leading to an ever-increasing incidence of invasive fungal infections (IFI). Due to the limited antifungal treatment options, the management of IFI remains a major challenge. The triazole antifungal drug isavuconazole (ISV) shows a broader spectrum of activity against Mucorales isolates and represents another therapeutic option for difficult-to-treat IFI. ISV is a broad-spectrum triazole antifungal II. generation, which is primarily intended for the treatment of invasive aspergillosis and mucormycosis, but in the future it also represents a promising therapeutic option for the treatment of other, rare IFIs (cryptococcosis, infections caused by dimorphic fungi). The article summarizes the basic knowledge and provides a brief overview of the pharmacodynamics, pharmacokinetics, mechanism of action, metabolism, indications, and dosage of isavuconazole in clinical practice. It also includes a brief analysis of selected clinical trials (SECURE, ACTIVE, VITAL) and recommendations of individual international societies.

MeSH Term

Pyridines
Nitriles
Triazoles
Humans
Invasive Fungal Infections
Antifungal Agents
Mucormycosis

Chemicals

isavuconazole
Pyridines
Nitriles
Triazoles
Antifungal Agents

Word Cloud

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